Fluconazole and Glimepiride: Drug Interaction Guide
Quick answer: This combination requires caution. Fluconazole and Glimepiride can be used together with adjustments and monitoring.
How Fluconazole interacts with Glimepiride
Fluconazole inhibits CYP2C9-mediated metabolism of glimepiride, increasing plasma levels and the risk of prolonged hypoglycaemia.
What you should do
Monitor capillary glucose closely and consider a 25–50% reduction of sulfonylurea dose during fluconazole therapy.
Key facts
Severity
Moderate — caution required
Mechanism
Fluconazole inhibits CYP2C9-mediated metabolism of glimepiride, increasing plasma levels and the risk of prolonged hypog...
Action
Monitor capillary glucose closely and consider a 25–50% reduction of sulfonylurea dose during fluconazole therapy.
Frequently asked questions
Can I take Fluconazole and Glimepiride together?
With caution. Monitor capillary glucose closely and consider a 25–50% reduction of sulfonylurea dose during fluconazole therapy.
What is the severity of this interaction?
The interaction between Fluconazole and Glimepiride is classified as Moderate — caution required. Fluconazole inhibits CYP2C9-mediated metabolism of glimepiride, increasing plasma levels and the risk of prolonged hypoglycaemia.
What should I do if I'm prescribed both?
Monitor capillary glucose closely and consider a 25–50% reduction of sulfonylurea dose during fluconazole therapy. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.