St John S Wort and Warfarin: Drug Interaction Guide
Quick answer: This combination requires caution. St John S Wort and Warfarin can be used together with adjustments and monitoring.
How St John S Wort interacts with Warfarin
St John's wort induces CYP3A4, CYP2C9, and P-glycoprotein through pregnane X receptor activation. This can reduce warfarin exposure and lower INR.
What you should do
Avoid St John's wort in patients taking warfarin. If started or stopped, monitor INR closely and adjust warfarin as needed.
Key facts
Severity
Moderate — caution required
Mechanism
St John's wort induces CYP3A4, CYP2C9, and P-glycoprotein through pregnane X receptor activation. This can reduce warfar...
Action
Avoid St John's wort in patients taking warfarin. If started or stopped, monitor INR closely and adjust warfarin as need...
Frequently asked questions
Can I take St John S Wort and Warfarin together?
With caution. Avoid St John's wort in patients taking warfarin. If started or stopped, monitor INR closely and adjust warfarin as needed.
What is the severity of this interaction?
The interaction between St John S Wort and Warfarin is classified as Moderate — caution required. St John's wort induces CYP3A4, CYP2C9, and P-glycoprotein through pregnane X receptor activation. This can reduce warfarin exposure and lower INR.
What should I do if I'm prescribed both?
Avoid St John's wort in patients taking warfarin. If started or stopped, monitor INR closely and adjust warfarin as needed. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.