Amiodarone and Dabigatran: Drug Interaction Guide
Quick answer: This is a major interaction — avoid combining Amiodarone and Dabigatran unless specifically directed by your doctor.
How Amiodarone interacts with Dabigatran
Amiodarone inhibits P-glycoprotein (P-gp) efflux transporter in the gut and kidney, increasing dabigatran absorption and reducing its renal clearance, leading to elevated plasma concentrations and bleeding risk.
What you should do
Reduce dabigatran dose to 110 mg twice daily when co-administered, especially in patients with CrCl 30–50 mL/min. Monitor for bleeding signs and consider alternative anticoagulation in elderly patients.
Key facts
Severity
Major — avoid combination
Mechanism
Amiodarone inhibits P-glycoprotein (P-gp) efflux transporter in the gut and kidney, increasing dabigatran absorption and...
Action
Reduce dabigatran dose to 110 mg twice daily when co-administered, especially in patients with CrCl 30–50 mL/min. Monito...
Frequently asked questions
Can I take Amiodarone and Dabigatran together?
No — this combination should generally be avoided. Reduce dabigatran dose to 110 mg twice daily when co-administered, especially in patients with CrCl 30–50 mL/min. Monitor for bleeding signs and consider alternative anticoagulation in elderly patients.
What is the severity of this interaction?
The interaction between Amiodarone and Dabigatran is classified as Major — avoid combination. Amiodarone inhibits P-glycoprotein (P-gp) efflux transporter in the gut and kidney, increasing dabigatran absorption and reducing its renal clearance, leading to elevated plasma concentrations and bleeding risk.
What should I do if I'm prescribed both?
Reduce dabigatran dose to 110 mg twice daily when co-administered, especially in patients with CrCl 30–50 mL/min. Monitor for bleeding signs and consider alternative anticoagulation in elderly patients. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.