Cyclosporine and Verapamil: Drug Interaction Guide
Quick answer: This combination requires caution. Cyclosporine and Verapamil can be used together with adjustments and monitoring.
How Cyclosporine interacts with Verapamil
Verapamil inhibits CYP3A4 and P-glycoprotein, reducing cyclosporine clearance. Cyclosporine exposure may increase, raising nephrotoxicity and hypertension risk.
What you should do
Monitor cyclosporine trough concentrations, renal function, and blood pressure; adjust cyclosporine dose as needed.
Key facts
Severity
Moderate — caution required
Mechanism
Verapamil inhibits CYP3A4 and P-glycoprotein, reducing cyclosporine clearance. Cyclosporine exposure may increase, raisi...
Action
Monitor cyclosporine trough concentrations, renal function, and blood pressure; adjust cyclosporine dose as needed.
Frequently asked questions
Can I take Cyclosporine and Verapamil together?
With caution. Monitor cyclosporine trough concentrations, renal function, and blood pressure; adjust cyclosporine dose as needed.
What is the severity of this interaction?
The interaction between Cyclosporine and Verapamil is classified as Moderate — caution required. Verapamil inhibits CYP3A4 and P-glycoprotein, reducing cyclosporine clearance. Cyclosporine exposure may increase, raising nephrotoxicity and hypertension risk.
What should I do if I'm prescribed both?
Monitor cyclosporine trough concentrations, renal function, and blood pressure; adjust cyclosporine dose as needed. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.