Amlodipine and Ciclosporin: Drug Interaction Guide
Quick answer: This combination requires caution. Amlodipine and Ciclosporin can be used together with adjustments and monitoring.
How Amlodipine interacts with Ciclosporin
Ciclosporin inhibits CYP3A4 metabolism of amlodipine, increasing plasma levels and risk of hypotension and peripheral oedema.
What you should do
Initiate amlodipine at low dose (2.5 mg) and titrate cautiously. Monitor blood pressure and watch for oedema; consider alternative antihypertensive.
Key facts
Severity
Moderate — caution required
Mechanism
Ciclosporin inhibits CYP3A4 metabolism of amlodipine, increasing plasma levels and risk of hypotension and peripheral oe...
Action
Initiate amlodipine at low dose (2.5 mg) and titrate cautiously. Monitor blood pressure and watch for oedema; consider a...
Frequently asked questions
Can I take Amlodipine and Ciclosporin together?
With caution. Initiate amlodipine at low dose (2.5 mg) and titrate cautiously. Monitor blood pressure and watch for oedema; consider alternative antihypertensive.
What is the severity of this interaction?
The interaction between Amlodipine and Ciclosporin is classified as Moderate — caution required. Ciclosporin inhibits CYP3A4 metabolism of amlodipine, increasing plasma levels and risk of hypotension and peripheral oedema.
What should I do if I'm prescribed both?
Initiate amlodipine at low dose (2.5 mg) and titrate cautiously. Monitor blood pressure and watch for oedema; consider alternative antihypertensive. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.