Paroxetine and Tramadol: Drug Interaction Guide
Quick answer: This is a major interaction — avoid combining Paroxetine and Tramadol unless specifically directed by your doctor.
How Paroxetine interacts with Tramadol
Paroxetine inhibits CYP2D6, the enzyme that converts tramadol to its active opioid metabolite (O-desmethyltramadol), reducing analgesia while serotonergic effects of both drugs combine to risk serotonin syndrome.
What you should do
Avoid combination; use a non-CYP2D6 dependent analgesic (e.g. paracetamol or morphine) and monitor for tremor, hyperreflexia and agitation.
Key facts
Severity
Major — avoid combination
Mechanism
Paroxetine inhibits CYP2D6, the enzyme that converts tramadol to its active opioid metabolite (O-desmethyltramadol), red...
Action
Avoid combination; use a non-CYP2D6 dependent analgesic (e.g. paracetamol or morphine) and monitor for tremor, hyperrefl...
Frequently asked questions
Can I take Paroxetine and Tramadol together?
No — this combination should generally be avoided. Avoid combination; use a non-CYP2D6 dependent analgesic (e.g. paracetamol or morphine) and monitor for tremor, hyperreflexia and agitation.
What is the severity of this interaction?
The interaction between Paroxetine and Tramadol is classified as Major — avoid combination. Paroxetine inhibits CYP2D6, the enzyme that converts tramadol to its active opioid metabolite (O-desmethyltramadol), reducing analgesia while serotonergic effects of both drugs combine to risk serotonin syndrome.
What should I do if I'm prescribed both?
Avoid combination; use a non-CYP2D6 dependent analgesic (e.g. paracetamol or morphine) and monitor for tremor, hyperreflexia and agitation. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.