Everolimus and Verapamil: Drug Interaction Guide

Quick answer: This is a major interaction — avoid combining Everolimus and Verapamil unless specifically directed by your doctor.

Interaction severity: Major — avoid combination

How Everolimus interacts with Verapamil

Verapamil inhibits CYP3A4 and P-glycoprotein, increasing everolimus exposure and risk of toxicity including stomatitis, pneumonitis and myelosuppression.

What you should do

Avoid combination if possible; if required, reduce everolimus dose and monitor trough concentrations and adverse effects closely.

Key facts

Severity

Major — avoid combination

Mechanism

Verapamil inhibits CYP3A4 and P-glycoprotein, increasing everolimus exposure and risk of toxicity including stomatitis, ...

Action

Avoid combination if possible; if required, reduce everolimus dose and monitor trough concentrations and adverse effects...

Important medical disclaimer: This page provides educational information about drug interactions for general reference. It is not a substitute for professional medical advice, diagnosis, or treatment. Always discuss your specific medications with a qualified healthcare provider before starting, stopping, or changing any treatment. About our editorial team.

Frequently asked questions

Can I take Everolimus and Verapamil together?

No — this combination should generally be avoided. Avoid combination if possible; if required, reduce everolimus dose and monitor trough concentrations and adverse effects closely.

What is the severity of this interaction?

The interaction between Everolimus and Verapamil is classified as Major — avoid combination. Verapamil inhibits CYP3A4 and P-glycoprotein, increasing everolimus exposure and risk of toxicity including stomatitis, pneumonitis and myelosuppression.

What should I do if I'm prescribed both?

Avoid combination if possible; if required, reduce everolimus dose and monitor trough concentrations and adverse effects closely. Always consult your prescribing clinician — do not stop or change medications without medical guidance.

Last reviewed: by iMedic Medical Editorial Team. Our editorial process.