Ciclosporin and Colchicine: Drug Interaction Guide
Quick answer: This is a major interaction — avoid combining Ciclosporin and Colchicine unless specifically directed by your doctor.
How Ciclosporin interacts with Colchicine
Ciclosporin inhibits P-glycoprotein and CYP3A4, markedly increasing colchicine exposure and risk of myopathy, neuropathy, and bone marrow toxicity.
What you should do
Avoid the combination, especially in renal or hepatic impairment. If essential, use specialist dosing advice and monitor for colchicine toxicity.
Key facts
Severity
Major — avoid combination
Mechanism
Ciclosporin inhibits P-glycoprotein and CYP3A4, markedly increasing colchicine exposure and risk of myopathy, neuropathy...
Action
Avoid the combination, especially in renal or hepatic impairment. If essential, use specialist dosing advice and monitor...
Frequently asked questions
Can I take Ciclosporin and Colchicine together?
No — this combination should generally be avoided. Avoid the combination, especially in renal or hepatic impairment. If essential, use specialist dosing advice and monitor for colchicine toxicity.
What is the severity of this interaction?
The interaction between Ciclosporin and Colchicine is classified as Major — avoid combination. Ciclosporin inhibits P-glycoprotein and CYP3A4, markedly increasing colchicine exposure and risk of myopathy, neuropathy, and bone marrow toxicity.
What should I do if I'm prescribed both?
Avoid the combination, especially in renal or hepatic impairment. If essential, use specialist dosing advice and monitor for colchicine toxicity. Always consult your prescribing clinician — do not stop or change medications without medical guidance.
Last reviewed: by iMedic Medical Editorial Team. Our editorial process.